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E-raamat: Advanced Pharmaceutical Solids

(University of Wisconsin (Emeritus), Madison, USA)
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This extensive reference/text explores the principles, instrumentation, processes, and programs of pharmaceutical solid science as well as new aspects on one-component systems, micromeritics, polymorphism, solid-state stability, cohesion, powder flow, blending, single- unit sustained release, and tablet coating. Reveals unique approaches in pharmaceutical solid science not previously published in any other text! Providing current data on crystallization, dissolution from particles and polydisperse populations, powder volumes and densities, comminution, wet granulation, and hard-shell capsules, Advanced Pharmaceutical Solids

describes moisture isotherms with crystalline solids

documents the effects of moisture on solid-state stability

highlights tablet physics and principles

explains sustained release by microencapsulation

presents prediction equations for solubility in binary solvents

discusses particle sizes and diameters

identifies Brunauer, Emmett, and Teller Isotherms

and more! Considering properties of solids, permeamitry and gas absorption methods, amorphates, and purification by pH-change precipitation, Advanced Pharmaceutical Solids is an essential reference for pharmacists; pharmaceutical scientists; medicinal, physical, surface, colloid, and analytical chemists and biochemists; and an effective text for upper-level undergraduate and graduate students in these disciplines.

Arvustused

" a comprehensive overview. "-Pharma Times

"would find good use as a textbook in a graduate level course on pharmaceutical solidsequally valuable as an information source for anyone seeking a brief overview of a particular area. "-Pharmaceutical Development Technology

"deserves a place on the bookshelves of any pharmaceutical scientist working on the development of solid dosage forms. an excellent initial reference for advanced students and scientists working on solids. "-Pharmaceutical Research

Preface v
One Component Systems
1(12)
Properties of Solids
13(14)
Solubility
27(24)
Particle Sizes and Diameters
51(10)
Micromeritics
61(28)
Crystallization
89(18)
Amorphates
107(10)
Polymorphism
117(16)
Moisture Isotherms with Crystalline Solids
133(26)
Drug Substance Considerations
159(10)
Melting Point Diagrams and Eutectics
169(22)
Dissolution from Particles and Surfaces
191(18)
Dissolution from Polydisperse Populations
209(14)
Solid State Stability
223(44)
Effect of Moisture on Solid-State Stability
267(14)
Apparent Volumes and Densities
281(18)
Cohesion
299(10)
Powder Flow
309(14)
Comminution
323(12)
Blending
335(18)
Wet Granulation
353(22)
Hard Shell Capsules
375(12)
Tablet Physics
387(20)
Physical Principles of Tablets
407(20)
Disintegration and Dissolution
427(12)
Polymers
439(16)
Coating of Tablets
455(14)
Single Unit Sustained Release Dosage Forms
469(24)
Sustained Release by Microencapsulation
493(18)
Index 511


Jens T. Carstensen